Absorption, Metabolism and Excretion of 14C-olorofim in Man

Sponsor
F2G Ltd
Study ID
NCT04039880
Phase
PHASE1
Status
Completed

Conditions

  • Invasive Fungal Infections

Eligibility Criteria

Sex
MALE
Age
18 Years - 55 Years
Healthy Volunteers
Accepted

Interventions

  • Olorofim — DRUG
    single oral dose (120 mg, 3.7 MBq)

Study Details

Single-centre, open-label, non-randomised, single dose study in 2 cohorts of healthy subjects. It is planned to enrol 6 healthy male subjects in Cohort A (standard mass balance and metabolite profiling cohort) and up to 6 subjects in Cohort B (biliary evaluation cohort); each subject will receive a single oral administration of 120 mg \[14C\]-olorofim oral solution containing approximately 3.7 MBq (100 µCi).

Key Dates

Start date
Jul 30, 2019
Status verified
Aug 2019
Primary completion
Sep 30, 2019
Completion
Sep 30, 2019

Study Design

Enrollment
12 participants (actual)
Allocation
NON_RANDOMIZED
Intervention model
SEQUENTIAL
Primary purpose
OTHER

Arms

  • Experimental: Cohort A (mass balance)
    evaluation of mass balance and metabolite profiling
  • Experimental: Cohort B (biliary evaluation)
    evaluation of biliary elimination

Primary Outcome Measure

Mass balance [ Time Frame: 28 days ]