A Study to Assess Naporafenib (ERAS-254) Administered With Trametinib in Patients With NRAS-mutant Melanoma (SEACRAFT-2)

Part of paid clinical trials in Phoenix, Arizona.

Sponsor
Erasca, Inc.
Study ID
NCT06346067
Phase
PHASE3
Status
Active Not Recruiting

Conditions

  • Advanced or Metastatic NRAS-mutant Melanoma

Eligibility Criteria

Sex
ALL
Age
18 Years - 99 Years
Healthy Volunteers
Not accepted

Interventions

  • Naporafenib — DRUG
    Naporafenib (ERAS-254) is an experimental Pan-Raf inhibitor
  • Dacarbazine — DRUG
    Dacarbazine IV - Day 1
  • Temozolomide — DRUG
    Temozolomide 200 mg/m2/day PO on Day 1 to Day 5 of each 28-day cycle
  • Trametinib — DRUG
    Trametinib is an FDA approved anticancer medication that targets MEK1 and MEK2.

Study Details

Stage 1: To select the optimal dose of naporafenib + trametinib to be studied in Stage 2. Stage 2: To compare progression free survival (PFS) and overall survival (OS) for patients with NRAS-mutant (NRASm) melanoma who are randomized to receive the combination of naporafenib + trametinib to that of patients who are randomized to physician's choice of therapy (dacarbazine, temozolomide, or trametinib monotherapy).

Key Dates

Start date
Apr 29, 2024
Status verified
Feb 2026
Primary completion
Apr 30, 2028
Completion
Dec 31, 2028

Study Design

Enrollment
78 participants (actual)
Allocation
RANDOMIZED
Intervention model
PARALLEL
Primary purpose
TREATMENT

Arms

  • Experimental: Stage 1 Dose selection Lead-in Arm 1
    Naporafenib + Trametinib Naporafenib (ERAS-254) 100 mg administered orally twice daily (BID) Trametinib 1 mg once daily (QD)
  • Experimental: Stage 1 Dose selection Lead-in Arm 2
    Naporafenib + Trametinib Naporafenib (ERAS-254) 400 mg administered orally twice daily (BID) Trametinib 0.5 mg once daily (QD)
  • Active Comparator: Stage 1 Dose selection Lead-in Arm 3 Trametinib monotherapy
    Trametinib 2 mg once daily (QD)
  • Experimental: Stage 2 Arm A
    Naporafenib + Trametinib Naporafenib (ERAS-254) BID oral administration with Trametinib QD at the dose selected in Stage 1
  • Active Comparator: Stage 2 Arm B - Physician's Choice
    * Dacarbazine 1000 mg/m2 intravenously (IV) on Day 1 of each 21-day cycle OR * Temozolomide 200 mg/m2/day PO on Day 1 to Day 5 of each 28-day cycle OR * Trametinib monotherapy, 2 mg PO QD

Primary Outcome Measure

Stage 1:To select the optimal dose of naporafenib + trametinib to be studied in Stage 2 [ Time Frame: Assessed up to 6 months from time of first dose ]

Locations (21)

FacilityCityStateZIPSite coordinators
Mayo Clinic - ArizonaPhoenixArizona85054-
University of California, San FranciscoSan FranciscoCalifornia94143-
The Melanoma and Skin Care InstituteEnglewoodColorado80113-
Mayo Clinic - FloridaJacksonvilleFlorida70121-
University of Miami Sylvester CancerMiamiFlorida33136-
University of Kansas Cancer CenterKansas CityKansas66205-
Ochsner Clinic FoundationJeffersonLouisiana70121-
Massachusetts General HospitalBostonMassachusetts02114-
Barbara Ann Karmanos Cancer InstituteDetroitMichigan48201-
Mayo ClinicRochesterMinnesota70121-
Washington University School of MedicineSt LouisMissouri63110-
Memorial Sloan Kettering Cancer CenterNew YorkNew York10065-
Cleveland Clinic FoundationClevelandOhio44195-
SCRI Oncology Partners (formerly Tennessee Oncology)NashvilleTennessee37203-
Texas Oncology- Austin MidtownAustinTexas78705-
Texas Oncology - Baylor Charles A. Sammons Cancer CenterDallasTexas75246-
The University of Texas MD Anderson Cancer CenterHoustonTexas77030-
The University of Utah - Huntsman Cancer Institute (HCI)Salt Lake CityUtah84112-
Virginia Oncology AssociatesNorfolkVirginia23502-1871-
Fred Hutchinson Cancer CenterSeattleWashington98109-
University of WisconsinMadisonWisconsin53792-

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